Objective: Study simple method to synthesis the α-arbutin for use in cosmetics. Method: We do respond glycosylated under Konigs-Knorr method improvements suggested by Helferich entire acetylated OH groups of glucose molecules and then conducted in response to monoacetyl glycosylated hydroquinone and then supply the hydrolysis protection group to obtain arbutin The reaction was examined under different conditions (temperature, time, catalyst gase environment...).