list of adrenergic drugs list of adrenergic drugs this is a list of adrenergic drugs. these are pharmaceutical drugs, naturally occurring compounds and other chemicals that influence the function of the neurotransmitter epinephrine (adrenaline). epinephrine receptor ligands agonists etilefrine amidephrine anisodamine anisodine cirazoline dipivefrine dopamine ephedrine epinephrine (adrenaline) etilefrine ethylnorepinephrine 5-fluoronorepinephrine 6-fluoronorepinephrine indanidine levonordefrin metaraminol methoxamine methyldopa midodrine naphazoline norepinephrine (noradrenaline) octopamine oxymetazoline phenylephrine phenylpropanolamine pseudoephedrine synephrine tetrahydrozoline antagonists abanoquil adimolol ajmalicine alfuzosin amosulalol arotinolol atiprosin benoxathian buflomedil bunazosin carvedilol ci-926 corynanthine dapiprazole dl-017 domesticine doxazosin eugenodilol fenspiride gyki-12,743 gyki-16,084 indoramin ketanserin l-765,314 labetalol mephendioxan metazosin monatepil moxisylyte (thymoxamine) naftopidil nantenine neldazosin nicergoline niguldipine pelanserin phendioxan phenoxybenzamine phentolamine piperoxan prazosin quinazosin ritanserin rs-97,078 sgb-1,534 silodosin sl-89.0591 spiperone talipexole tamsulosin terazosin tibalosin tiodazosin tipentosin tolazoline trimazosin upidosin urapidil zolertine many tricyclic antidepressants, tetracyclic antidepressants, antipsychotics, ergolines, and some piperazines like buspirone, trazodone, nefazodone, etoperidone, and mepiprazole antagonize α1-adrenergic receptors as well, which contributes to their side effects such as orthostatic hypotension. agonists adrenoswitches (photoswitchable agonists) amitraz apraclonidine brimonidine cannabivarin clonidine detomidine dexmedetomidine dihydroergotamine dipivefrine dopamine ephedrine ergotamine epinephrine (adrenaline) esproquin etilefrine ethylnorepinephrine 6-fluoronorepinephrine guanabenz guanfacine guanoxabenz levonordefrin lofexidine medetomidine methyldopa mivazerol naphazoline 4-nemd (r)-3-nitrobiphenyline norepinephrine (noradrenaline) phenylpropanolamine piperoxan pseudoephedrine rilmenidine romifidine talipexole tetrahydrozoline tizanidine tolonidine urapidil xylazine xylometazoline antagonists adimolol aptazapine atipamezole brl-44408 buflomedil cirazoline efaroxan esmirtazapine fenmetozole fluparoxan gyki-12,743 gyki-16,084 idazoxan mianserin mirtazapine mk-912 nan-190 olanzapine phentolamine phenoxybenzamine piperoxan piribedil pyrimidinylpiperazine rauwolscine rotigotine sb-269,970 setiptiline spiroxatrine sunepitron tolazoline yohimbine many atypical antipsychotics and azapirones like buspirone and gepirone (via metabolite pyrimidinylpiperazine) antagonize α2-adrenergic receptors as well. agonists salbutamol abediterol amibegron arbutamine arformoterol arotinolol bambuterol befunolol bitolterol bromoacetylalprenololmenthane (baam) broxaterol buphenine carbuterol cimaterol clenbuterol denopamine deterenol dipivefrine dobutamine dopamine dopexamine ephedrine epinephrine (adrenaline) etafedrine etilefrine ethylnorepinephrine fenoterol 2-fluoronorepinephrine 5-fluoronorepinephrine formoterol hexoprenaline higenamine indacaterol isoetarine isoprenaline (isoproterenol) n-isopropyloctopamine isoxsuprine labetalol levonordefrin levosalbutamol mabuterol methoxyphenamine methyldopa norepinephrine (noradrenaline) orciprenaline oxyfedrine phenylpropanolamine pirbuterol prenalterol ractopamine procaterol pseudoephedrine quinterenol reproterol rimiterol ritodrine salbutamol (albuterol) salmeterol solabegron terbutaline tretoquinol tulobuterol xamoterol zilpaterol zinterol antagonists acebutolol adaprolol adimolol afurolol alprenolol alprenoxime amosulalol ancarolol arnolol arotinolol atenolol befunolol betaxolol bevantolol bisoprolol bopindolol bornaprolol brefonalol bucindolol bucumolol bufetolol bufuralol bunitrolol bunolol bupranolol butaxamine butidrine butofilolol capsinolol carazolol carpindolol carteolol carvedilol celiprolol cetamolol cicloprolol cinamolol cloranolol cyanopindolol dalbraminol dexpropranolol diacetolol dichloroisoprenaline dihydroalprenolol dilevalol diprafenone draquinolol ecastolol epanolol ericolol ersentilide esatenolol esmolol eugenodilol exaprolol falintolol flestolol flusoxolol hydroxycarteolol hydroxytertatolol ici-118,551 idropranolol indenolol indopanolol iodocyanopindolol iprocrolol isoxaprolol isamoltane labetalol landiolol levobetaxolol levobunolol levocicloprolol levomoprolol medroxalol mepindolol metalol metipranolol metoprolol moprolol nadolol nadoxolol nafetolol nebivolol neraminol nifenalol nipradilol oberadilol oxprenolol pacrinolol pafenolol pamatolol pargolol parodilol penbutolol penirolol phqa-33 pindolol pirepolol practolol primidolol procinolol pronethalol propafenone propranolol ridazolol ronactolol soquinolol sotalol spirendolol sr 59230a sulfinalol ta-2005 talinolol tazolol teoprolol tertatolol tienoxolol tilisolol timolol tiprenolol tolamolol toliprolol tribendilol trigevolol xibenolol xipranolol reuptake inhibitors norepinephrine transporter (net) inhibitors reboxetine selective norepinephrine reuptake inhibitors amedalin atomoxetine (tomoxetine) ciclazindol daledalin esreboxetine lortalamine mazindol nisoxetine reboxetine talopram talsupram tandamine viloxazine norepinephrine-dopamine reuptake inhibitors amineptine bupropion (amfebutamone) fencamine fencamfamine lefetamine levophacetoperane lr-5182 manifaxine methylphenidate nomifensine o-2172 radafaxine serotonin-norepinephrine reuptake inhibitors bicifadine desvenlafaxine duloxetine eclanamine levomilnacipran milnacipran sibutramine venlafaxine serotonin-norepinephrine-dopamine reuptake inhibitors brasofensine diclofensine dov-102,677 dov-21,947 dov-216,303 jnj-7925476 jz-iv-10 methylnaphthidate naphyrone ns-2359 prc200-ss sep-225,289 sep-227,162 tesofensine tricyclic antidepressants amitriptyline butriptyline cianopramine clomipramine desipramine dosulepin doxepin imipramine lofepramine melitracen nortriptyline protriptyline trimipramine tetracyclic antidepressants amoxapine maprotiline mianserin oxaprotiline setiptiline others cocaine cp-39,332 exp-561 fezolamine ginkgo biloba indeloxazine nefazodone nefopam pridefrine tapentadol teniloxazine tramadol ziprasidone vesicular monoamine transporter (vmat) inhibitors ibogaine reserpine tetrabenazine bietaserpine releasing agents aminorex morpholines fenbutrazate morazone phendimetrazine phenmetrazine oxazolines aminorex clominorex cyclazodone fenozolone fluminorex 4-methylaminorex pemoline thozalinone phenethylamines (also amphetamines, cathinones, phentermines, etc.) 2-oh-pea 4-cab 4-fa 4-fma 4-ma 4-mma alfetamine amfecloral amfepentorex amfepramone amphetamine dextroamphetamine levoamphetamine amphetaminil β-me-pea bdb benzphetamine boh buphedrone butylone cathine cathinone clobenzorex clortermine d-deprenyl dimethylamphetamine dimethylcathinone (dimethylpropion, metamfepramone) dma dmma ebdb ephedrine ethcathinone ethylamphetamine ethylone famprofazone fenethylline fenproporex flephedrone fludorex furfenorex hordenine iap imp lisdexamfetamine lophophine mbdb mda (tenamfetamine) mdea mdma mdmpea mdoh mdpea mefenorex mephedrone mephentermine methamphetamine dextromethamphetamine levomethamphetamine methcathinone methedrone methylone nap ortetamine paredrine pba pca pentorex (phenpentermine) phenethylamine pholedrine phenpromethamine phentermine phenylpropanolamine pia prenylamine propylamphetamine pseudoephedrine selegiline (l-deprenyl) tiflorex tyramine xylopropamine zylofuramine piperazines benzylpiperazine (bzp) 2,5-dimethoxy-4-bromobenzylpiperazine (2c-b-bzp) methylbenzylpiperazine (mbzp) metachlorophenylpiperazine (mcpp) methylenedioxybenzylpiperazine (mdbzp) methoxyphenylpiperazine (meopp) parafluorophenylpiperazine (pfpp) others 2-amino-1,2-dihydronaphthalene 2-aminoindane 2-aminotetralin 2-benzylpiperidine 4-benzylpiperidine clofenciclan cyclopentamine cypenamine cyprodenate feprosidnine gilutensin heptaminol hexacyclonate indanorex 5-iodo-2-aminoindane (5-iai) isometheptene methylhexanamine octodrine phthalimidopropiophenone propylhexedrine levopropylhexedrine tuaminoheptane enzyme inhibitors phenylalanine hydroxylase (pah) inhibitors 3,4-dihydroxystyrene tyrosine hydroxylase inhibitors 3-iodotyrosine aquayamycin bulbocapnine metirosine oudenone aromatic l-amino acid decarboxylase (aaad) inhibitors benserazide carbidopa genistein methyldopa dopamine-beta-hydroxylase (dbh) inhibitors bupicomide disulfiram dopastin fusaric acid nepicastat phenopicolinic acid tropolone phenylethanolamine n-methyltransferase (pnmt) inhibitors cgs-19281a skf-64139 skf-7698 monoamine oxidase (mao) inhibitors selegiline nonselective benmoxin caroxazone echinopsidine furazolidone hydralazine indantadol iproclozide iproniazid isocarboxazid isoniazid linezolid mebanazine metfendrazine nialamide octamoxin paraxazone phenelzine pheniprazine phenoxypropazine pivalylbenzhydrazine procarbazine safrazine tranylcypromine mao-a selective amiflamine bazinaprine befloxatone befol brofaromine cimoxatone clorgiline esuprone harmala alkaloids harmine harmaline tetrahydroharmine harman norharman etc. methylene blue metralindole minaprine moclobemide pirlindole sercloremine tetrindole toloxatone tyrima mao-b selective d-deprenyl selegiline (l-deprenyl) ladostigil lazabemide milacemide mofegiline pargyline rasagiline safinamide mao-b inhibitors also influence norepinephrine/epinephrine levels since they inhibit the breakdown of their precursor dopamine. catechol-o-methyl transferase (comt) inhibitors entacapone tolcapone others precursors l-phenylalanine l-phenylalanine → l-tyrosine → l-dopa (levodopa) → dopamine l-dops (droxidopa) cofactors ferrous iron (fe2+) s-adenosyl-l-methionine vitamin b3 niacin nicotinamide → nadph vitamin b6 (pyridoxine, pyridoxamine, pyridoxal → pyridoxal phosphate) vitamin b9 (folic acid → tetrahydrofolic acid) vitamin c ascorbic acid zinc (zn2+) activity enhancers benzofuranylpropylaminopentane (bpap) phenylpropylaminopentane (ppap) release blockers bethanidine bretylium guanadrel guanazodine guanclofine guanethidine guanoxan toxins oxidopamine (6-hydroxydopamine)